Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04684
Ion Channel
Sodium channel protein type 9 subunit alpha
Peptide Function
Blocker
Gene Name
Scn9a
Activity Data (nM)
IC50
177000 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
KWDRDHKR
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
[CHEMBL1917113; BDBM50357365]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available
Experimental Conditions
pH
Not mention
Holding Potential (mV)
−100 mV
Temperature
∼21 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available